Table 2. A typical experiment aimed at the detection of the modulating effect of a small compound (SC) on kinetics (affinity) of binary BBI .
Panel |
Protein analyte * (µM) / SC (µM) |
|||||
Reference |
0.01 / 0 |
0.05 / 0 |
0.1 / 0 |
0.5 / 0 |
1 / 0 |
10 / 0 |
Control |
0 / 10 |
0 / 25 |
0 / 50 |
0 / 75 |
0 / 100 |
0 / 200 |
Targeted №1 |
0.01 / 10 |
0.05 / 10 |
0.1 / 10 |
0.5 / 10 |
1 / 10 |
10 / 10 |
Targeted №2 |
0.01 / 25 |
0.05 / 25 |
0.1 / 25 |
0.5 / 25 |
1 / 25 |
10 / 25 |
Targeted №3 |
0.01 / 50 |
0.05/ 50 |
0.1 / 50 |
0.5 / 50 |
1 / 50 |
10 / 50 |
Targeted №4 |
0.01/ 75 |
0.05 / 75 |
0.1 / 75 |
0.5 / 75 |
1 / 75 |
10 / 75 |
Targeted №5 |
0.01/ 100 |
0.05 / 100 |
0.1 / 100 |
0.5 / 100 |
1 / 100 |
10 / 100 |
Targeted №6 |
0.01 / 200 |
0.05/ 200 |
0.1 / 200 |
0.5 / 200 |
1 / 200 |
10 / 200 |
Note. *Protein analyte was injected to the cell in solution while its partner (protein ligand) was covalently immobilized onto an optical biosensor chip.